"Relaxon" preparation: instructions for use, description, reviews, analogues

In what dose is the preparation "Relaxon" prescribed? Instructions for use of the medicament will be discussed below. Also you will learn about whether there are analogues for this medicine, how much it costs, in what cases it is not prescribed, etc.

Form, description, composition and packaging

The preparation "Relaxon" is available in the form of round biconvex tablets of white color,covered with a film sheath. The active substance of this drug is zopiclone. Also in the composition of the medicament are the following auxiliary substances: methyloxypropylcellulose, microcrystalline cellulose, lactose, potato starch, colloidal silicon dioxide, talc, sodium carboxymethyl starch, povidone, macrogol, magnesium stearate and titanium dioxide.

In what kind of packaging are the tablets "Relaxon" sold? Instructions for use are enclosed in a pack of cardboard, where the contour cells with the drug are placed.

Pharmacodynamic characteristics of

How does the Relaxone drug work? Instruction for use reports that this is a hypnotic, belonging to the group of cyclopirrolone. Structurally, it differs from barbiturates and hypnotic benzodiazepine series. This drug is a benzodiazepine receptor agonist. Interacting with them, it does not come into contact with peripheral receptors.

Properties of the preparation

What are the properties of the "Relaxon" medication? Experts say that this tool is able to have sedative, moderate anticonvulsant sleeping pills, muscle relaxant and tranquilizing effects. All of them are related to the action from the receptors of the macromolecular complex GABA.

After taking the pill, the inhibitory effect of GABA is increased, and the interneuronal transmission to the central nervous system is suppressed.

Sleeping "Relaxon" significantly shortens the time of falling asleep, reduces the number of awakenings at night and improves the quality of sleep. Also this drug increases the duration of sleep and almost does not cause such post-somnical effects as drowsiness and malaise in the morning.

There is no adaptation to the drug. Therefore, it can be taken in a batch mode up to 17 weeks.

Pharmacokinetics of the drug

The drug "Relaxon", the price of which is indicated below, is quickly absorbed and is observed in the blood after 2 hours. The intake of food does not affect the absorption of the drug in any way. At 45%, it binds to blood proteins.

Even after several pills, the accumulation of their active substance, as well as metabolites, is not noted.

The half-life of zopiclone and the main metabolites is 7.5 and 4.5 hours, and the unchanged zopiclone is 5.5 hours. Approximately 80% of the drug is excreted together by urine, and 17-20% with feces.

In elderly people, the metabolism of the drug in the liver is somewhat reduced. At the same time, its half-life is extended to 7 hours. As for the accumulation of the active substance, it is not detected with repeated administration of tablets.

Indications for use

What to do with insomnia? Doctors recommend taking "Relaxon".This drug is designed to treat chronic, situational and transient insomnia in adults. Also it is actively used by those who have difficulty with falling asleep, early and night awakenings.

Contraindications to the use of

Tablets "Relaxon" is not recommended in the following cases:

• with increased sensitivity to the main substance of the medication;
• in severe myasthenia gravis;
• during pregnancy;
• for sleep apnea;
• with respiratory failure;
• for severe hepatic insufficiency;
• under the age of 18 years.

The preparation "Relaxon": instructions for use

It is recommended to consult a doctor before taking a sleeping pill. Also it is necessary to study the attached instruction.

Tablets "Relaxon"( international name - "Zopiclone") are taken orally, shortly before the onset of sleep. Adults receive this medication at a dose of 7.5 mg. The maximum amount of sleeping pills is 15 mg.

The total duration of the use of tablets should not be more than one month. In each individual case, the duration of therapy is determined individually, depending on the patient's condition and the form of insomnia.

To take the drug with transient insomnia, it is desirable about 3-5 days, and for a situational - 2.5-3 weeks. The duration of the course therapy for chronic insomnia should be determined only by the doctor.

Elderly people with chronic pulmonary insufficiency, as well as with impaired liver function, are prescribed 3.75 mg of the drug. If necessary, this dosage may be increased to 7.5 mg.

Treatment of insomnia in patients with kidney failure also begin with ½ tablets, that is, with 3.75 mg.

Cases of overdose

Taking large doses of hypnotics causes CNS depression of varying severity( from pronounced drowsiness to coma).

Overdose therapy starts with a gastric lavage. Then the patient is assigned sorbents.

Symptomatic treatment and monitoring of vital body functions is also carried out. The drug "Flumazenil" is used as an antidote.

Side effects of

What are the side effects of Relaxon? The responses of experienced specialists report that this medication can contribute to the development of the following phenomena:

• nausea, dryness and bitterness in the mouth;
• dizziness, headache, minor morning drowsiness;
• nightmares, aggressiveness, irritability, hallucinations, mood deterioration and depressive state, as well as the development of amnesia( very rarely);
• itching, the appearance of rash, anaphylactic reactions( extremely rare);
• increased liver transaminases and alkaline phosphatase.

It should also be noted that in rare cases, the drug causes the "cancellation" syndrome and as a consequence, ricochet insomnia.

Drug Interaction

Now you know what to do with insomnia. Reception of the drug "Relaxon" should be extremely cautious, especially with the simultaneous use of other medications.

According to the attached instructions, the intensification of the oppressive effect on the CNS of this drug occurs when combined with antidepressants, neuroleptics, anesthetics, tranquilizers, sedatives and hypnotics, as well as "Erythromycin", antiepileptic and antihistamines, narcotic analgesics.

It is highly not recommended to drink alcoholic beverages and alcohol-containing medicines at the same time as Relaxon. This is due to the fact that such a combination can enhance its sedative effect.

Taking a hypnotic drug markedly reduces the concentration of perforanal or trimipramine in the blood. This fact should be taken into account when they are simultaneously assigned.

Special recommendations for taking a sleeping pill

What should I know before taking Relaxon( analogs of this remedy are listed below)?

In people with nocturnal seizures of bronchial asthma in combination with medications of the methylxanthine series, the hypnotic reduces the number of attacks in the pre-hours, and also reduces their intensity and duration.

When appointing Relaxon, you should not completely exclude the possibility of developing addiction. The risk of dependence on the drug occurs in the following cases:

• if the duration of treatment and dosage is impaired;
• for the abuse of alcoholic beverages or other medicines;
• when combined with alcohol or other psychotropic drugs.

To avoid the syndrome of "cancellation", stop taking medication gradually, reducing the dosage to a minimum.

When taking sleeping pills, the patient may experience anterograde amnesia. As a rule, it manifests itself in the interruption of sleep, and after a long time between taking the medication and going to sleep.

To reduce such risks, it is necessary: ​​

• to provide a sleep duration of at least 6 hours;
• take the medicine just before bedtime.

This medication is not indicated for depression therapy. He can mask her symptoms.

An effective and safe dose of "Relaxon" in children and adolescents under 18 years has not been established by specialists. Therefore, taking the drug at this age is prohibited.

Due to the pharmacological properties of the hypnotic, it can adversely affect a patient's ability to drive vehicles, as well as engage in hazardous activities that require increased attention and quick response. In this regard, during the treatment with this drug should be extremely cautious.

Sleeping "Relaxon": price and analogues

What can I replace the drug "Relaxon"?This drug has many analogues. The most effective are the following medications: Milovan, Imovan, Thorson, Somnol, Slipwell, Zolinox, Piklodorm, Zopiclone.

All listed products, including "Relaxon", are dispensed in pharmacies only on the prescription of a doctor. As for the price, this means it is not very high.20 tablets of sleeping pills( 7.5 mg) can be purchased for 120-160 rubles.

Reviews of sleeping pills

According to specialists, the drug "Relaxon" is a sleeping drug of the third generation. By the way, they include Zaleplon and Zolpidem. These drugs are highly effective and absolutely safe.

Patients report that, after taking sleeping pills, their sleep quality has improved markedly. At the same time, the fast-phase sleep, necessary for restoring the psycho-emotional state, was completely preserved.

This medication has a good effect on the slow-wave phase of sleep, which is extremely important for the physical recovery of the human body.

According to specialists, this drug contributes to the normalization of the structure of sleep in all types of disorders. At the same time, it has the least likelihood of addiction.

The patient's testimonies indicate that the sleeping pills "Relaxon" are well tolerated, without having any effect on the person's daily activity. However, doctors do not recommend taking this medicine on your own. The patient should always consult a doctor and follow all the recommended dosages.